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Research ArticleCancer
Synergistic action of the MCL-1 inhibitor S63845 with current therapies in preclinical models of triple-negative and HER2-amplified breast cancer
- View ORCID ProfileDelphine Merino1,2,*,
- View ORCID ProfileJames R. Whittle1,2,3,*,
- View ORCID ProfileFrançois Vaillant1,2,*,
- Antonin Serrano1,2,
- View ORCID ProfileJia-Nan Gong2,4,
- Goknur Giner2,5,
- Ana Leticia Maragno6,
- Maïa Chanrion6,
- Emilie Schneider6,
- Bhupinder Pal1,2,
- Xiang Li2,7,
- Grant Dewson2,7,
- Julius Gräsel1,2,
- Kevin Liu1,2,
- View ORCID ProfileNajoua Lalaoui2,7,
- David Segal2,4,
- Marco J. Herold2,8,
- View ORCID ProfileDavid C. S. Huang2,4,
- View ORCID ProfileGordon K. Smyth5,9,
- Olivier Geneste6,
- View ORCID ProfileGuillaume Lessene2,10,11,
- View ORCID ProfileJane E. Visvader1,2,† and
- Geoffrey J. Lindeman1,3,12,13,†
- 1ACRF Stem Cells and Cancer Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
- 2Department of Medical Biology, University of Melbourne, Parkville, Victoria 3010, Australia.
- 3Department of Medical Oncology, Peter MacCallum Cancer Centre, Melbourne, Victoria 3000, Australia.
- 4Cancer and Haematology Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
- 5Bioinformatics Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
- 6Institut de Recherches Servier Oncology R&D Unit, Croissy Sur Seine 78290, France.
- 7Cell Signalling and Cell Death Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
- 8Molecular Genetics of Cancer Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
- 9School of Mathematics and Statistics, University of Melbourne, Parkville, Victoria 3010, Australia.
- 10Chemical Biology Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
- 11Department of Pharmacology and Therapeutics, University of Melbourne, Parkville, Victoria 3010, Australia.
- 12Department of Medicine, University of Melbourne, Parkville, Victoria 3010, Australia.
- 13Parkville Familial Cancer Centre, Royal Melbourne Hospital and Peter MacCallum Cancer Centre, Parkville, Victoria 3050, Australia.
- ↵†Corresponding author. Email: visvader{at}wehi.edu.au (J.E.V.); lindeman{at}wehi.edu.au (G.J.L.)
↵* These authors contributed equally to this work.
See allHide authors and affiliations
Science Translational Medicine 02 Aug 2017:
Vol. 9, Issue 401, eaam7049
DOI: 10.1126/scitranslmed.aam7049
Vol. 9, Issue 401, eaam7049
DOI: 10.1126/scitranslmed.aam7049
Delphine Merino
1ACRF Stem Cells and Cancer Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
2Department of Medical Biology, University of Melbourne, Parkville, Victoria 3010, Australia.
James R. Whittle
1ACRF Stem Cells and Cancer Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
2Department of Medical Biology, University of Melbourne, Parkville, Victoria 3010, Australia.
3Department of Medical Oncology, Peter MacCallum Cancer Centre, Melbourne, Victoria 3000, Australia.
François Vaillant
1ACRF Stem Cells and Cancer Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
2Department of Medical Biology, University of Melbourne, Parkville, Victoria 3010, Australia.
Antonin Serrano
1ACRF Stem Cells and Cancer Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
2Department of Medical Biology, University of Melbourne, Parkville, Victoria 3010, Australia.
Jia-Nan Gong
2Department of Medical Biology, University of Melbourne, Parkville, Victoria 3010, Australia.
4Cancer and Haematology Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
Goknur Giner
2Department of Medical Biology, University of Melbourne, Parkville, Victoria 3010, Australia.
5Bioinformatics Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
Ana Leticia Maragno
6Institut de Recherches Servier Oncology R&D Unit, Croissy Sur Seine 78290, France.
Maïa Chanrion
6Institut de Recherches Servier Oncology R&D Unit, Croissy Sur Seine 78290, France.
Emilie Schneider
6Institut de Recherches Servier Oncology R&D Unit, Croissy Sur Seine 78290, France.
Bhupinder Pal
1ACRF Stem Cells and Cancer Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
2Department of Medical Biology, University of Melbourne, Parkville, Victoria 3010, Australia.
Xiang Li
2Department of Medical Biology, University of Melbourne, Parkville, Victoria 3010, Australia.
7Cell Signalling and Cell Death Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
Grant Dewson
2Department of Medical Biology, University of Melbourne, Parkville, Victoria 3010, Australia.
7Cell Signalling and Cell Death Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
Julius Gräsel
1ACRF Stem Cells and Cancer Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
2Department of Medical Biology, University of Melbourne, Parkville, Victoria 3010, Australia.
Kevin Liu
1ACRF Stem Cells and Cancer Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
2Department of Medical Biology, University of Melbourne, Parkville, Victoria 3010, Australia.
Najoua Lalaoui
2Department of Medical Biology, University of Melbourne, Parkville, Victoria 3010, Australia.
7Cell Signalling and Cell Death Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
David Segal
2Department of Medical Biology, University of Melbourne, Parkville, Victoria 3010, Australia.
4Cancer and Haematology Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
Marco J. Herold
2Department of Medical Biology, University of Melbourne, Parkville, Victoria 3010, Australia.
8Molecular Genetics of Cancer Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
David C. S. Huang
2Department of Medical Biology, University of Melbourne, Parkville, Victoria 3010, Australia.
4Cancer and Haematology Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
Gordon K. Smyth
5Bioinformatics Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
9School of Mathematics and Statistics, University of Melbourne, Parkville, Victoria 3010, Australia.
Olivier Geneste
6Institut de Recherches Servier Oncology R&D Unit, Croissy Sur Seine 78290, France.
Guillaume Lessene
2Department of Medical Biology, University of Melbourne, Parkville, Victoria 3010, Australia.
10Chemical Biology Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
11Department of Pharmacology and Therapeutics, University of Melbourne, Parkville, Victoria 3010, Australia.
Jane E. Visvader
1ACRF Stem Cells and Cancer Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
2Department of Medical Biology, University of Melbourne, Parkville, Victoria 3010, Australia.
Geoffrey J. Lindeman
1ACRF Stem Cells and Cancer Division, Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria 3052, Australia.
3Department of Medical Oncology, Peter MacCallum Cancer Centre, Melbourne, Victoria 3000, Australia.
12Department of Medicine, University of Melbourne, Parkville, Victoria 3010, Australia.
13Parkville Familial Cancer Centre, Royal Melbourne Hospital and Peter MacCallum Cancer Centre, Parkville, Victoria 3050, Australia.
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