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Research ArticleCancer
A rationally designed NRP1-independent superagonist SEMA3A mutant is an effective anticancer agent
- Noemi Gioelli1,2,*,
- Federica Maione2,3,*,
- Chiara Camillo1,2,
- Michela Ghitti4,
- Donatella Valdembri1,2,
- Noemi Morello5,
- Marie Darche6,
- Lorena Zentilin7,
- Gabriella Cagnoni1,2,
- Yaqi Qiu2,3,
- Mauro Giacca7,
- Maurizio Giustetto5,8,
- Michel Paques9,10,
- Ilaria Cascone6,
- Giovanna Musco4,
- Luca Tamagnone1,2,†,
- Enrico Giraudo2,3,†,‡ and
- Guido Serini1,2,†,‡
- 1Department of Oncology, University of Torino School of Medicine, 10060 Candiolo, Torino, Italy.
- 2Candiolo Cancer Institute, FPO-IRCCS, 10060 Candiolo, Torino, Italy.
- 3Department of Science and Drug Technology, University of Torino, 10125 Torino, Italy.
- 4Biomolecular NMR Unit, IRCCS Ospedale San Raffaele, 20132 Milano, Italy.
- 5Department of Neuroscience, University of Torino School of Medicine, 10126 Torino, Italy.
- 6Growth, Reparation and Tissue Regeneration Laboratory, ERL-CNRS 9215, University of Paris-Est, 94000 Créteil, France.
- 7Molecular Medicine Laboratory, International Centre for Genetic Engineering and Biotechnology, 34149 Trieste, Italy.
- 8National Institute of Neuroscience-Italy, 10126 Torino, Italy.
- 9Vision Institute, Sorbonne University, UPMC University of Paris 06, INSERM, CNRS, 75012 Paris, France.
- 10Centre Hospitalier National d’Ophtalmologie des Quinze-Vingts, INSERM-DHOS CIC 503, 75012 Paris, France.
- ↵‡Corresponding author. Email: guido.serini{at}ircc.it (G.S.); enrico.giraudo{at}ircc.it (E.G.)
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Science Translational Medicine 23 May 2018:
Vol. 10, Issue 442, eaah4807
DOI: 10.1126/scitranslmed.aah4807
Vol. 10, Issue 442, eaah4807
DOI: 10.1126/scitranslmed.aah4807
Noemi Gioelli
Department of Oncology, University of Torino School of Medicine, 10060 Candiolo, Torino, Italy.Candiolo Cancer Institute, FPO-IRCCS, 10060 Candiolo, Torino, Italy.
Federica Maione
Candiolo Cancer Institute, FPO-IRCCS, 10060 Candiolo, Torino, Italy.Department of Science and Drug Technology, University of Torino, 10125 Torino, Italy.
Chiara Camillo
Department of Oncology, University of Torino School of Medicine, 10060 Candiolo, Torino, Italy.Candiolo Cancer Institute, FPO-IRCCS, 10060 Candiolo, Torino, Italy.
Michela Ghitti
Biomolecular NMR Unit, IRCCS Ospedale San Raffaele, 20132 Milano, Italy.
Donatella Valdembri
Department of Oncology, University of Torino School of Medicine, 10060 Candiolo, Torino, Italy.Candiolo Cancer Institute, FPO-IRCCS, 10060 Candiolo, Torino, Italy.
Noemi Morello
Department of Neuroscience, University of Torino School of Medicine, 10126 Torino, Italy.
Marie Darche
Growth, Reparation and Tissue Regeneration Laboratory, ERL-CNRS 9215, University of Paris-Est, 94000 Créteil, France.
Lorena Zentilin
Molecular Medicine Laboratory, International Centre for Genetic Engineering and Biotechnology, 34149 Trieste, Italy.
Gabriella Cagnoni
Department of Oncology, University of Torino School of Medicine, 10060 Candiolo, Torino, Italy.Candiolo Cancer Institute, FPO-IRCCS, 10060 Candiolo, Torino, Italy.
Yaqi Qiu
Candiolo Cancer Institute, FPO-IRCCS, 10060 Candiolo, Torino, Italy.Department of Science and Drug Technology, University of Torino, 10125 Torino, Italy.
Mauro Giacca
Molecular Medicine Laboratory, International Centre for Genetic Engineering and Biotechnology, 34149 Trieste, Italy.
Maurizio Giustetto
Department of Neuroscience, University of Torino School of Medicine, 10126 Torino, Italy.National Institute of Neuroscience-Italy, 10126 Torino, Italy.
Michel Paques
Vision Institute, Sorbonne University, UPMC University of Paris 06, INSERM, CNRS, 75012 Paris, France.Centre Hospitalier National d’Ophtalmologie des Quinze-Vingts, INSERM-DHOS CIC 503, 75012 Paris, France.
Ilaria Cascone
Growth, Reparation and Tissue Regeneration Laboratory, ERL-CNRS 9215, University of Paris-Est, 94000 Créteil, France.
Giovanna Musco
Biomolecular NMR Unit, IRCCS Ospedale San Raffaele, 20132 Milano, Italy.
Luca Tamagnone
Department of Oncology, University of Torino School of Medicine, 10060 Candiolo, Torino, Italy.Candiolo Cancer Institute, FPO-IRCCS, 10060 Candiolo, Torino, Italy.
Enrico Giraudo
Candiolo Cancer Institute, FPO-IRCCS, 10060 Candiolo, Torino, Italy.Department of Science and Drug Technology, University of Torino, 10125 Torino, Italy.
Guido Serini
Department of Oncology, University of Torino School of Medicine, 10060 Candiolo, Torino, Italy.Candiolo Cancer Institute, FPO-IRCCS, 10060 Candiolo, Torino, Italy.
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